Cart
sales@molnova.com
EPZ 025654
CAS No. 1888328-89-9
EPZ 025654 ( EPZ025654;EPZ-025654;GSK 35336023 )
Catalog No. M12957 CAS No. 1888328-89-9
EPZ025654 (GSK 35336023) is a potent, selective arginine methyltransferase CARM1 inhibitor with IC50 of 3 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 1413 | Get Quote |
|
| 50MG | 2862 | Get Quote |
|
| 100MG | 3870 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
-
Product NameEPZ 025654
-
NoteResearch use only, not for human use.
-
Brief DescriptionEPZ025654 (GSK 35336023) is a potent, selective arginine methyltransferase CARM1 inhibitor with IC50 of 3 nM.
-
DescriptionEPZ025654 (GSK 35336023) is a potent, selective arginine methyltransferase CARM1 inhibitor with IC50 of 3 nM.
-
SynonymsEPZ025654;EPZ-025654;GSK 35336023
-
PathwayChromatin/Epigenetic
-
TargetHMTase
-
RecptorHMTase
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number1888328-89-9
-
Formula Weight577.09
-
Molecular FormulaC29H33ClN8O3
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESO[C@H](CNC)COC1=CC=C(Cl)C(C2=NC(C3=C(C)ON=C3C)=C(C)C(N4CC5=NC(N6CCC6)=NC=C5C4)=N2)=C1
-
Chemical Name(R)-1-(3-(4-(2-(azetidin-1-yl)-5,7-dihydro-6H-pyrrolo[3,4-d]pyrimidin-6-yl)-6-(3,5-dimethylisoxazol-4-yl)-5-methylpyrimidin-2-yl)-4-chlorophenoxy)-3-(methylamino)propan-2-ol
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Drew AE, et al. Sci Rep. 2017 Dec 21;7(1):17993.
molnova catalog
related products
-
UNC-1079
The piperidine analog of UNC1021; structurally similar but significantly less potent inhibitor for use as a negative control in cellular studies.
-
MI-2-2
MI-2-2 is a potent inhibitor of the menin-MLL interaction that binds to menin with low nanomolar affinity (Kd=22 nM).
-
HLCL-61 hydrochlorid...
A novel potent and selective protein arginine methyltransferase PRMT5 inhibitor.
